1995

  • M. Gairí, P. Lloyd- Williams, F. Albericio, E. Giralt.
    Convergent solid-phase peptide synthesis. 12* Chromatographic techniques for the purification of protected peptide segments. Int. J. Peptide Protein Res., 46, 119-133. (1995).
  • I. Dalcol, F. Rabanal, M-D Ludevid, F. Albericio and E. Giralt.
    Convergent Solid Phase Peptide Synthesis: An Efficient Approach to the Synthesis of Highly Repetitive Protein Domains. J. Org. Chem., 60, 7575-7581 (1995).
  • E. Nicolás, M. Vilaseca and E. Giralt.
    A study of the use of NH4I for the reduction of methionine sulfoxide in peptides containing cysteine and cystine. Tetrahedron, 51, 5701-5710 (1995).
  • N. Verdaguer, M. Mateu, E. Giralt, D. Andreu, E. Domingo and I. Fita.
    Structure of the major 1antigenic loop of foot-and-mouth disease virus complexed with a neutralizing antibody: direct involvement of the Arg-Gly-Asp motif in the interaction. EMBO J., 14, 1690-1696 (1995).
  • A. Adeva, J. Camarero, E. Giralt and D. Andreu.
    Boc S-methylbenzyl-(S)-2-amino-6-mercaptohexanoic acid: Preparation and application to the synthesis of a large cyclic disulfide peptide. Tetrahedron Lett., 36, 3885-3888 (1995).
  • J. Camarero, E. Giralt and D. Andreu.
    Cyclization of a large disulfide peptide in the solid phase. Tetrahedron Lett., 36, 1137-1140 (1995).
  • M-L Valero, J. Camarero, A. Adeva, N. Verdaguer, I. Fita, M. Mateu, E. Domingo, E. Giralt and D. Andreu. Cyclic peptides as conformationally restricted models of viral antigens. Application to foot-and-mouth disease virus. Biomed. Pept. Prot. Nucl. Acids, 1, 133-140 (1995).
  • M. Royo, J. Alsina, E. Giralt, U. Slomcyznska and F. Albericio.
    S-Phenylacetamidomethyl (Phacm): an orthogonal cysteine protecting group for Boc and Fmoc solid-phase peptide synthesis strategies. J. Chem. Soc. Perkin Trans. I, 1095-1102 (1995).
  • F. Rabanal, E. Giralt and F. Albericio.
    Synthesis and applications of a new base-labile fluorene derived linker for solid-phase peptide synthesis. Tetrahedron, 51, 1449-1458 (1995).
  • J. Camarero, J. Cairó, E. Giralt and D. Andreu.
    Solution versus solid-phase cyclization strategies for large sidechain lactam-bridged peptides: a comparative study. J. Peptide Sci., 1, 241-250 (1995).
  • E. Crusi, E. Giralt and D. Andreu.
    Peptide ionophores: Synthesis and cation-binding properties of a bicyclic peptide containing glycine and lysine residues. Peptide Res., 8, 62-69 (1995).
  • M. Mateu, J. Camarero, E. Giralt, D. Andreu and E. Domingo.
    Direct evaluation of the immunodominance of a major antigenic site of foot-and-mouth disease virus in a natural host. Virology, 206, 298-306 (1995).
  • E. Nicolas, J. Bacardit, T. Ferrer, E. Giralt.
    CD studies of peptides that mimic the four helicoidal sequences of the uteroglobin sp; monomer. Lett. in Peptide Science, 2, 353-362. (1995).
  • J.A. Camarero, A. Adeva, M.G. Mateu, E. Domingo, E. Giralt, D. Andreu.
    Cyclic peptide mimetics of the major antigenic site of foot-and-mouth disease virus. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 857-858 (1995).
  • C. Carreño, A.L. Carrascosa, E. Viñuela, E. Giralt, D. Andreu.
    A synthetic analog of African swine fever virus p12 attachment factor: The redesign of a synthetically difficult protein. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 807-808 (1995).
  • E. Nicolás, J. Bacardit, M. Vilaseca, E. Giralt.
    C.D. studies of uteroglobin fragments. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 570-571 (1995).
  • F. Albericio, J. Bacardit, G. Barany, J.M. Coull, M. Egholm, E. Giralt, G.W. Griffin, S.S. Kates, E. Nicolás, N.A. Solé.
    Polyethylene glycol-polystryrene (PEG-PS) supports for Boc solid-phase peptide and PNA synthesis strategies. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 271-272 (1995).
  • F. Alberico, I. Abdelmoty, J. Bofill, L. Carpino, A. El-Faham, B. Foxman, M. Gairí, E. Giralt, G. Griffin, S. Kates, P. Lloyd-Williams, C. Minor, L. Scarmoutzos, H. Shroff, S. Triolo and H. Wenschuh. Azabenzotriazole (HOAt) derivatives as superior coupling reagents for peptide synthesis. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium" (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 23-25.(1995).
  • P. LLoyd-Williams, P. Monerris, I. Gonzalez, G. Jou, E. Giralt.
    Synthesis of D-allo-isoleucine from L-isoleucine and from (S)-2-methyl-1-butanol:Synthesis of isostatine. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 209-210 (1995).
  • M. Royo, F. Albericio, E. Giralt, M. Pons.
    Helicity and superhelicity in cyclic coiled-coil peptides. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 83-84 (1995).
  • I. Dalcol, F. Rabanal, F. Albericio, M. Pons, M. Geli, M. Torrent, M.D. Ludevid, E. Giralt.
    A proline-rich region from maize Y-zein adopts a left-handed amphipathic structure that may act as a signal for its retention in the endoplasmic reticulum. In "Peptides 1994. Proceedings of the Twenty-Third European Peptide Symposium". (H.L.S. Maia, ed.), Escom, Science Publishers, Leiden, The Netherlands, 1995, pp. 60-61 (1995).

1996

  • E. Domingo, M. G. Mateu, C. Escarmis, E. Martínez-Salas, D. Andreu, E. Giralt, N. Verdaguer and I. Fita. Molecular Evolution of Aphthoviruses. Virus Genes, 11, 197-207, (1996).
  • R. Rodríguez, I. Viñets, A. Diez, M. Rubiralta and E. Giralt.
    Conformationally Restricted Analogues of Tryptophan: Synthesis of Chiral 3-Amino-4-Indolyl-2-Piperidones. Synthetic Communications, 26, 3029-3059 (1996).
  • I. Dalcol, M. Pons, M-D. Ludevid and E. Giralt.
    Convergent Synthesis of Repeating Peptides (Val-X-Leu-Pro-Pro-Pro)8 Adopting a Polyproline II Conformation. J. Org. Chem., 61, 6775-6782 (1996).
  • J. Alsina, E. Giralt and F. Albericio.
    Use of N-Tritylamino Acids and PyAOP1 for the Suppression of Diketopiperazine Formation in Fmoc/tBu Solid-Phase Peptide Synthesis Using Alkoxybenzyl Ester Anchoring Linkages. Tetrahedron Letters, 37, 4195-4198 (1996).
  • D. Andreu, J.A. Camarero, M.L. Valero, X. Roig, T. Haack, E. Giralt, N. Verdaguer, I. Fita, M.G. Mateu and E. Domingo.
    Synthetic, Structural and Immunochemical Approaches to Antigen-Antibody Interactions in Foot-and-Mouth Disease Virus. In "Peptides, Chemistry, Structure and Biology. Procedings of the Fourteenth American Peptide Symposium". (Pravin T. P. Kaumaya and Robert S. Hodges, eds), Mayflower Scientific Ltd., pp. 875-877 (1996).
  • Y.M. Sánchez, T. Haack, M.J. González, D. Ludevid, E. Giralt.
    Is the Topological Equivalence Between Retro-enantiomers a General Concept? In "Peptides, Chemistry, Structure and Biology. Procedings of the Fourteenth American Peptide Symposium". (Pravin T. P. Kaumaya and Robert S. Hodges, eds), Mayflower Scientific Ltd., pp. 558-560. (1996).
  • I. González, G. Jou, J. M. Caba, F. Albericio, P. Lloyd-Williams, E. Giralt.
    Synthesis of derivatives of (2S,4S)-4-hydroxy-2,5-dimethyl-3-oxohexanoic acid, a constituent of the didemnins. J. Chem. Soc. Perkin Trans. I, 1427-1433 (1996).
  • M.L. Valero, E. Giralt, D. Andreu.
    Solid Phase-Mediated Cyclization of Head-to-Tail Peptides: Problems Associated with Slide Chain Anchoring. Tetrahedron Lett., 37, 4229-4232 (1996).
  • C. Alemán, A. M. Ilarduya, E. Giralt, S. Muñóz-Guerra.
    Analysis of the Conformational Preferences of (4R,5R)-4,5-Bis(alkylcarbamoyl)-1,3-dioxolanes. Tetrahedron, 24, 8275-8286 (1996).
  • G. Guichard, S. Muller, M. Regenmortel, J.P. Briand, P. Mascagni, E. Giralt.
    Structural limitations to antigenic mimicry achievable with retroinverso (all-D-retro) peptides. TIBTECH, 14, 44-45 (1996).
  • R. Rodríguez, A. Diez, M. Rubiralta, E. Giralt.
    Synthesis of 3-Amino-4-Indolyl-2 Piperidones: Tryptophan -Derived Pseudodipeptides. Heterocycles, 43, 513-517 (1996).
  • J. Sánchez-Quesada, Ch. Seel, P. Prados, J. Mendoza, I. Dalcol, E. Giralt.
    Anion Helicates: Double Strand Helical Self-Assembly of Chiral Bicyclic Guanidinium Dimers and Tetramers around Sulfate Templates. J. Am. Chem. Soc., 118, 277-278 (1996).

1997

  • T. Haack, Mª J.González, Y. Sánchez and E. Giralt.
    D-Amino Acids in protein de novo design II. Protein-Diastereomerism versus Protein Enantiomerism. Lett. in Peptide Science, 4, 1-10 (1997).
  • F. Albericio, P. Lloyd-Williams and E. Giralt.
    Convergent Solid-Phase Peptide Synthesis. In: "Methods in Enzymology" (Gregg B. Fields, ed.), Academic Press, 289, pp. 313-336 (1997).
  • N. Thieriet, J. Alsina, E. Giralt, F. Guibé and F. Albericio.
    Use of Alloc-amino Acids in Solid-Phase Peptide Synthesis. Tandem Deprotection-Coupling Reactions Using Neutral Conditions. Tetrahedron Lett., 38, 7275-7278 (1997).
  • M. Gairí, R. Romi, I. Fernández, H. Rochat, M-F. Martin, J. van Rietschoten, M. Pons and E. Giralt.
    3D Structure of Kaliotoxin: Is Residue 34 a Key for Channel Selectivity? J. Peptide Sci, 3, 314-319 (1997).
  • T. Haack, Y. Sánchez, M-J. González and E. Giralt.
    Structural Comparison in Solution of a Native and Retro Peptide Derived from the Third Helix of Staphylococcus aureus Protein A, Domain B: Retro Peptides, a Useful Tool for the Discrimination of Helix Stabilization Factors Dependent on the Peptide Chain Orientation. J. Peptide Sci, 3, 299-313 (1997).
  • M. W. Peczuh, A. D. Hamilton, J. Sánchez-Quesada, J. de Mendoza, T. Haack and E. Giralt.
    Recognition and Stabilization of an a-Helical Peptide by a Synthetic Receptor. J.Am. Chem. Soc., 119, 9327-9328 (1997).
  • T. Haack, J. Camarero, X. Roig, M. Mateu, E. Domingo, D. Andreu and E. Giralt.
    A cyclic disulfide peptide reproduces in solution the main structural features of a native antigenic site of foot-and-mouth disease virus. Int. J. Biol. Macromolecules, 20, 209-219 (1997).
  • P. Lloyd-Williams, F. Albericio, M. Gairí and E. Giralt.
    The purification of protected peptide segments. In: Innovation and Perspectives in Solid Phase Synthesis; Combinatorial Libraries. (Roger Epton, ed). Mayflower Scientific Ltd., pp. 195-200 (1997).
  • E. Nicolás, M. Pujades, J. Bacardit, E. Giralt and F. Albericio.
    A New Approach to Hmb-backbone Protection of Peptides: Synthesis and Reactivity of Na-Fmoc- Na-(Hmb)amino Acids1. Tetrahedron Lett., 38, 2317-2320 (1997).
  • O. Taboga, C. Tami, E. Carrillo, J. I. Nuñez, A. Rodríguez, J. C. Saiz, E. Blanco, M.L. Valero, X. Roig, J.A. Camarero, D. Andreu, M. G. Mateu, E. Giralt, E. Domingo, F. Sobrino, and E. Palma.
    A Large-Scale Evaluation of Peptide Vaccines against Foot-and-Mouth Disease: Lack of Solid Protectio in Cattle and Isolation of Escape Mutants. J. Virol., 71, 2606-2 614 (1997).
  • M.A. Contreras, T. Haack, M. Royo, E. Giralt and M. Pons.
    Temperature coefficients of peptides dissolved in hexafluoroisopropanol monitor distortions of helices. Lett. in Peptide Science, 4, 29-39 (1997).
  • C. Ibarra, R. Fernández, M. Quiroga, A. Carbonell, F. Cárdenas and E. Giralt.
    New Approach to Thiazolo[5,4-b]quinoline Derivatives, Synthesis, Cytotoxicity and DNA-Interaction. J. Med. Chem., 40, 668-676 (1997).
  • P. Lloyd-Williams, A. Sánchez, N. Carulla, T. Ochoa and E. Giralt.
    Synthetic Studies on Threonines. The Preparation of Protected Derivatives of D-allo-Threonine for Peptide Synthesis. Tetrahedron, 53, 3369-3382 (1997).
  • E. Nicolás, J. Clemente, T. Ferrer, F. Albericio and E. Giralt.
    The Use of the Nbb-Resin for the Solid-Phase Synthesis of Peptide Alkylesters and Alkylamides. Synthesis of Leuprolide. Tetrahedron Lett., 53, 3179-3194 (1997).
  • G. Jou, I. González, F. Albericio, P. Lloyd-Williams and E. Giralt.
    Total Synthesis of Dehydrodidemnim B. Use of Uronium and Phosphonium Salt Coupling Reagents in Peptide Synthesis in Solution. J. Org. Chem, 62, 354-366 (1997).
  • J. Alsina, C. Chiva, M. Ortiz, F. Rabanal, E. Giralt and F. Albericio.
    Active Carbonate Resins for Solid-Phase Synthesis Trough the Anchoring of a Hydroxyl Function. Synthesis of Cyclic and Alcohol Peptides. Tetrahedron Lett., 38, 883-886 (1997).
  • P. Lloyd-Williams, N. Carulla and E. Giralt.
    Simple Methods for the Preparation of Protected Derivatives of D-allo and L-allo -Threonine. Tetrahedron Lett., 38, 299-302 (1997).